Sexual HealthLimited Research⚠️ Not Approved — Caution

Melanotan II

MT-II · Non-selective melanocortin receptor agonism (MC1R, MC3R, MC4R, MC5R); MC1R activation produces melanin for tanning; MC4R activation causes penile erection and appetite suppression; lacks MC2R selectivity causing adrenal side effects

Not medical advice. For educational and research reference only.

Typical Dose

Research: 0.5–1 mg (extreme caution; not recommended)

Route

Injectable

Cycle

Not recommended for ongoing use

Storage

2–8°C Refrigerated

What is Melanotan II?

Melanotan II (MT-II) is a synthetic analog of α-melanocyte-stimulating hormone (α-MSH) studied for skin tanning, erectile function, and appetite suppression. Not FDA-approved and associated with significant safety concerns including dangerous nausea, uncontrolled melanocytic changes (nevi/moles), hypertension, and priapism. The FDA has issued multiple warnings. Banned from 503A compounding. Use with extreme caution.

Mechanism of Action

Non-selective melanocortin receptor agonism (MC1R, MC3R, MC4R, MC5R); MC1R activation produces melanin for tanning; MC4R activation causes penile erection and appetite suppression; lacks MC2R selectivity causing adrenal side effects

Target: MC1R, MC3R, MC4R, MC5R (non-selective)

Research Indications

Sexual FunctionEffective

Research and clinical data supporting effects on sexual response

Libido SupportEffective

Clinical data shows improvements in desire and arousal metrics

Melanocortin ActivityModerate

Acts via central nervous system melanocortin receptor pathways

Research Protocols

These are commonly discussed research protocols — not medical advice. Consult a healthcare provider before use.

GoalDoseFrequencyRoute
Starting DoseLow dosePer protocolVaries
Standard DoseTitratedPer protocolVaries

Peptide & Drug Interactions

Always consult your healthcare provider before combining with other compounds. Use our Interaction Checker for reference.

PDE5 Inhibitors (Sildenafil, Tadalafil)Monitor
Blood Pressure MedicationsCaution
Other Melanocortin AgonistsAvoid
NaltrexoneMonitor

How to Reconstitute & Inject

Use bacteriostatic (BAC) water only. Avoid saline — may cause precipitation. Refrigerate and use within 28 days.

  1. 1

    Remove Melanotan II vial from refrigeration and allow to reach room temperature (15–20 minutes)

  2. 2

    Clean vial top with alcohol swab and allow to air dry completely

  3. 3

    Using a sterile syringe, draw the calculated volume of bacteriostatic water (BAC water)

  4. 4

    Inject BAC water slowly down the side of the vial — do not aim directly at the powder

  5. 5

    Gently swirl in circular motions — DO NOT shake vigorously as this degrades the peptide

  6. 6

    Allow 2–3 minutes for full dissolution — solution should be clear and colorless

  7. 7

    Draw calculated dose into an insulin syringe for subcutaneous injection

  8. 8

    Inject into abdomen, thigh, or upper arm. Rotate injection sites to prevent lipodystrophy

  9. 9

    Store reconstituted solution refrigerated (2–8°C) and use within 28 days

What to Expect

Week 1–2

Initial effects and adaptation period. Monitor for any adverse reactions.

Week 2–4

Primary effects begin to manifest. Adjust dosing as recommended by your provider.

Week 4–8

Main therapeutic effects should be established. Assess progress with your provider.

Week 8+

Evaluate results and determine continuation, cycling, or dose adjustments.

Side Effects & Safety

  • Injection site reactions (redness, bruising, mild pain)
  • Potential for allergic reaction — discontinue if rash or hives occur
  • Individual reactions vary — start at the lowest dose and monitor carefully
  • Consult your healthcare provider before use and report any unusual symptoms

Melanotan II is banned from 503A compounding pharmacies. Only available through 503B outsourcing facilities or for research use.

FDA Status & Regulatory Info

⚠️ Not Approved — Caution

Melanotan II (MT-II) is a synthetic analog of α-melanocyte-stimulating hormone (α-MSH) studied for skin tanning, erectile function, and appetite suppression. Not FDA-approved and associated with significant safety concerns including dangerous nausea, uncontrolled melanocytic changes (nevi/moles), hypertension, and priapism. The FDA has issued multiple warnings. Banned from 503A compounding. Use with extreme caution.

Rx Required: No
503A Ban: Yes
Telehealth: N/A
Full FDA Status Tracker

Frequently Asked Questions

Research References

External links for education only. We do not control third-party content.

Community-reported data

The information below reflects self-reported experiences from PeptIQ app users. It is not clinical evidence and should not replace professional medical advice.

Community Intelligence

What 46 users report

46 community reports

Positive 97% · Neutral 3% · Negative 0%

Most reported benefits

Mood
142
Libido
142
Appetite
74

Most reported side effects

Fatigue
2
Nausea
2

Dose distribution

Median: 400–600 mcg · Most common: 200–400 mcg

0–25
1
25–50
0
50–100
1
100–200
7
200–400
48
400–600
23
600–1000
33
1000–2000
29
2000+
0

How repeat users are trending

Among repeat reporters, 94% said they felt similar to their last entry, 6% more positive, and 0% more negative.

Overall, repeat reporters leaned more positive than their previous entry.

Median gap between entries: 50 days · Based on 32 repeat reporters

Share Your Experience

Rate Melanotan II in the PeptIQ app and help the community make informed decisions.

Research purposes only

This page is for educational reference. It is not medical or legal advice. Consult the FDA and a licensed healthcare professional for current regulations and individualized guidance.