Immune SupportLimited ResearchResearch Only

KPV

α-MSH C-terminal tripeptide · MC1R and MC3R partial agonism; NF-κB nuclear translocation inhibition; direct intracellular uptake reducing pro-inflammatory cytokines (IL-1β, TNF-α, IL-8, IL-6); inhibition of caspase-1 and NLRP3 inflammasome activation

Not medical advice. For educational and research reference only.

Typical Dose

500 mcg–2 mg daily (research protocols)

Route

Injectable

Cycle

Protocol-dependent

Storage

2–8°C Refrigerated

What is KPV?

KPV is the C-terminal tripeptide (Lys-Pro-Val) of alpha-melanocyte stimulating hormone (α-MSH), retaining its potent anti-inflammatory properties without melanocortin receptor-dependent melanization effects. Research demonstrates significant potential for inflammatory bowel disease (IBD), Crohn's disease, skin inflammatory conditions, and wound healing. Oral formulations show promise for gut-specific delivery. Research only.

Mechanism of Action

MC1R and MC3R partial agonism; NF-κB nuclear translocation inhibition; direct intracellular uptake reducing pro-inflammatory cytokines (IL-1β, TNF-α, IL-8, IL-6); inhibition of caspase-1 and NLRP3 inflammasome activation

Target: MC1R, MC3R, NF-κB, NLRP3 inflammasome

Research Indications

Immune ModulationEffective

Research shows modulation of immune cell activity and inflammatory response

Inflammation ControlEffective

May reduce systemic and localized inflammatory markers

Infection ResistanceModerate

Some evidence for improved pathogen defense mechanisms

Research Protocols

These are commonly discussed research protocols — not medical advice. Consult a healthcare provider before use.

GoalDoseFrequencyRoute
Starting Dose250 mcg3x weeklySubcutaneous injection
Maintenance Dose500 mcgWeeklySubcutaneous injection

Peptide & Drug Interactions

Always consult your healthcare provider before combining with other compounds. Use our Interaction Checker for reference.

Consult prescriber before combining with any medicationCaution
BPC-157Compatible
NAD+Compatible
Vitamin DCompatible

How to Reconstitute & Inject

Use bacteriostatic (BAC) water only. Avoid saline — may cause precipitation. Refrigerate and use within 28 days.

  1. 1

    Remove KPV vial from refrigeration and allow to reach room temperature (15–20 minutes)

  2. 2

    Clean vial top with alcohol swab and allow to air dry completely

  3. 3

    Using a sterile syringe, draw the calculated volume of bacteriostatic water (BAC water)

  4. 4

    Inject BAC water slowly down the side of the vial — do not aim directly at the powder

  5. 5

    Gently swirl in circular motions — DO NOT shake vigorously as this degrades the peptide

  6. 6

    Allow 2–3 minutes for full dissolution — solution should be clear and colorless

  7. 7

    Draw calculated dose into an insulin syringe for subcutaneous injection

  8. 8

    Inject into abdomen, thigh, or upper arm. Rotate injection sites to prevent lipodystrophy

  9. 9

    Store reconstituted solution refrigerated (2–8°C) and use within 28 days

What to Expect

Week 1–2

Initial effects and adaptation period. Monitor for any adverse reactions.

Week 2–4

Primary effects begin to manifest. Adjust dosing as recommended by your provider.

Week 4–8

Main therapeutic effects should be established. Assess progress with your provider.

Week 8+

Evaluate results and determine continuation, cycling, or dose adjustments.

Side Effects & Safety

  • Injection site reactions (redness, bruising, mild pain)
  • Potential for allergic reaction — discontinue if rash or hives occur
  • Individual reactions vary — start at the lowest dose and monitor carefully
  • Consult your healthcare provider before use and report any unusual symptoms

FDA Status & Regulatory Info

Research Only

KPV is the C-terminal tripeptide (Lys-Pro-Val) of alpha-melanocyte stimulating hormone (α-MSH), retaining its potent anti-inflammatory properties without melanocortin receptor-dependent melanization effects. Research demonstrates significant potential for inflammatory bowel disease (IBD), Crohn's disease, skin inflammatory conditions, and wound healing. Oral formulations show promise for gut-specific delivery. Research only.

Rx Required: No
503A Ban: No
Telehealth: Available
Full FDA Status Tracker

Frequently Asked Questions

Research References

External links for education only. We do not control third-party content.

Community-reported data

The information below reflects self-reported experiences from PeptIQ app users. It is not clinical evidence and should not replace professional medical advice.

Community Intelligence

What 54 users report

54 community reports

Positive 98% · Neutral 2% · Negative 0%

Most reported benefits

Recovery
210
Mood
210

Dose distribution

Median: 200–400 mcg · Most common: 200–400 mcg

0–25
0
25–50
0
50–100
0
100–200
0
200–400
116
400–600
89
600–1000
3
1000–2000
1
2000+
1

How repeat users are trending

Among repeat reporters, 95% said they felt similar to their last entry, 5% more positive, and 0% more negative.

Overall, repeat reporters leaned more positive than their previous entry.

Median gap between entries: 60 days · Based on 43 repeat reporters

Share Your Experience

Rate KPV in the PeptIQ app and help the community make informed decisions.

Research purposes only

This page is for educational reference. It is not medical or legal advice. Consult the FDA and a licensed healthcare professional for current regulations and individualized guidance.