AntimicrobialLimited ResearchResearch Only

LL-37

Cathelicidin hCAP18 · Membrane disruption of microbial cells via electrostatic interaction with anionic phospholipids; TLR4 modulation and FPRL1 (formyl peptide receptor like-1) signaling for immune modulation; promotes keratinocyte migration and angiogenesis via EGF receptor transactivation

Not medical advice. For educational and research reference only.

Typical Dose

Research setting (doses not established for humans)

Route

Injectable

Cycle

Research protocol-dependent

Storage

2–8°C Refrigerated

What is LL-37?

LL-37 is the only cathelicidin antimicrobial peptide expressed in humans, derived from cleavage of the C-terminus of hCAP18. It demonstrates broad-spectrum antimicrobial activity against bacteria (including MRSA), fungi, and viruses, and also plays critical roles in wound healing, immune modulation, and anti-tumor activity. Expressed primarily in neutrophils, epithelial cells, and skin. Research only.

Mechanism of Action

Membrane disruption of microbial cells via electrostatic interaction with anionic phospholipids; TLR4 modulation and FPRL1 (formyl peptide receptor like-1) signaling for immune modulation; promotes keratinocyte migration and angiogenesis via EGF receptor transactivation

Target: Microbial membranes, TLR4, FPRL1, EGF receptor

Research Indications

Antimicrobial ActivityEffective

Demonstrated broad-spectrum antimicrobial properties in research

Wound Infection PreventionModerate

May help prevent microbial colonization of wounds

Immune ActivationModerate

Activates innate immune responses against pathogens

Research Protocols

These are commonly discussed research protocols — not medical advice. Consult a healthcare provider before use.

GoalDoseFrequencyRoute
Starting DoseLow dosePer protocolVaries
Standard DoseTitratedPer protocolVaries

Peptide & Drug Interactions

Always consult your healthcare provider before combining with other compounds. Use our Interaction Checker for reference.

Consult prescriber before combining with any medicationCaution
BPC-157Compatible
NAD+Compatible
Vitamin DCompatible

How to Reconstitute & Inject

Use bacteriostatic (BAC) water only. Avoid saline — may cause precipitation. Refrigerate and use within 28 days.

  1. 1

    Remove LL-37 vial from refrigeration and allow to reach room temperature (15–20 minutes)

  2. 2

    Clean vial top with alcohol swab and allow to air dry completely

  3. 3

    Using a sterile syringe, draw the calculated volume of bacteriostatic water (BAC water)

  4. 4

    Inject BAC water slowly down the side of the vial — do not aim directly at the powder

  5. 5

    Gently swirl in circular motions — DO NOT shake vigorously as this degrades the peptide

  6. 6

    Allow 2–3 minutes for full dissolution — solution should be clear and colorless

  7. 7

    Draw calculated dose into an insulin syringe for subcutaneous injection

  8. 8

    Inject into abdomen, thigh, or upper arm. Rotate injection sites to prevent lipodystrophy

  9. 9

    Store reconstituted solution refrigerated (2–8°C) and use within 28 days

What to Expect

Week 1–2

Initial effects and adaptation period. Monitor for any adverse reactions.

Week 2–4

Primary effects begin to manifest. Adjust dosing as recommended by your provider.

Week 4–8

Main therapeutic effects should be established. Assess progress with your provider.

Week 8+

Evaluate results and determine continuation, cycling, or dose adjustments.

Side Effects & Safety

  • Injection site reactions (redness, bruising, mild pain)
  • Potential for allergic reaction — discontinue if rash or hives occur
  • Individual reactions vary — start at the lowest dose and monitor carefully
  • Consult your healthcare provider before use and report any unusual symptoms

FDA Status & Regulatory Info

Research Only

LL-37 is the only cathelicidin antimicrobial peptide expressed in humans, derived from cleavage of the C-terminus of hCAP18. It demonstrates broad-spectrum antimicrobial activity against bacteria (including MRSA), fungi, and viruses, and also plays critical roles in wound healing, immune modulation, and anti-tumor activity. Expressed primarily in neutrophils, epithelial cells, and skin. Research only.

Rx Required: No
503A Ban: No
Telehealth: N/A
Full FDA Status Tracker

Frequently Asked Questions

Research References

External links for education only. We do not control third-party content.

Community-reported data

The information below reflects self-reported experiences from PeptIQ app users. It is not clinical evidence and should not replace professional medical advice.

Community Intelligence

What 6 users report

6 community reports

Positive 100% · Neutral 0% · Negative 0%

Most reported benefits

Recovery
6

Dose distribution

Median: 100–200 mcg · Most common: 100–200 mcg

0–25
0
25–50
0
50–100
0
100–200
4
200–400
2
400–600
0
600–1000
0
1000–2000
0
2000+
0

Commonly stacked with

Share Your Experience

Rate LL-37 in the PeptIQ app and help the community make informed decisions.

Research purposes only

This page is for educational reference. It is not medical or legal advice. Consult the FDA and a licensed healthcare professional for current regulations and individualized guidance.